TargetOther named receptors

Cholecystokinin receptor type A

A named receptor outside the families above. The catch-all is explicit rather than silent: these are receptors, but they are not grouped.

Measurements: 24
Compounds: 12
Binding constants: 7
Median pX: —

I · Identity

What this target is

Its function as UniProt states it, where in a cell the protein is found, and which cell types and tissues transcribe its gene.

Cholecystokinin receptor type A is a cell line or an assay label, not a protein, so there is no gene to describe. Its measurements are still shown below — they are real, and they are measurements of what a compound did in that system rather than of what it binds.

Resolver said a cell line or assay label, not a gene — recorded by tools/fetch_expression.py, not written here.

IV · Evidence

Every measurement at this target

Each row links to the ChEMBL assay it came from.

Equilibrium binding constants 7

Ki and Kd — a concentration at equilibrium. Directly comparable across rows at the same target.

Target	Class	Type	Value (nM)	pX	Organism	Assay
Cholecystokinin receptor type A	Other named receptors	Ki	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	Ki	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	Ki	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	Ki	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	Ki	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	Ki	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	Ki	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129

Functional readouts 17

IC₅₀, EC₅₀, AC₅₀ and potency. Assay-dependent, and not interchangeable with a binding constant.

Target	Class	Type	Value (nM)	pX	Organism	Assay
Cholecystokinin receptor type A	Other named receptors	IC50	34,000	4.47	Mus musculus	CHEMBL651446
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	IC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	IC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	IC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	IC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	IC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	IC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757
Cholecystokinin receptor type A	Other named receptors	IC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL1909129
Cholecystokinin receptor type A	Other named receptors	AC50	— no normalized value	— value does not convert to pX	Homo sapiens	CHEMBL5291757

← All targets