Plasma
Preparations such as liver microsomes or whole blood. Values below are reported as measured; because this is not a molecular target, they are not treated as affinities anywhere on this site.
- Measurements
- 10
- Compounds
- 3
- Binding constants
- 0
- Median pX
- —
I · Identity
What this target is
Its function as UniProt states it, where in a cell the protein is found, and which cell types and tissues transcribe its gene.
Plasma has no protein record here. A name resolves when ChEMBL’s own target record gives an accession, when the name appears verbatim in a gene’s synonym list, or when it matches a UniProt protein name exactly. Guessing from a name that merely looks like a receptor is how a histone gene ends up filed as an adrenoceptor.
IV · Evidence
Every measurement at this target
Each row links to the ChEMBL assay it came from.
Other measurements 10
Everything else ChEMBL recorded for this compound — percentage inhibition, efficacy, half-life, cytotoxicity. Reported in the assay's own units, which is why no value is converted here.
| Target | Class | Type | Value (nM) | pX | Organism | Assay |
|---|---|---|---|---|---|---|
| Plasma | Tissue and matrix | Fu | — no normalized value | — value does not convert to pX | Rattus norvegicus | CHEMBL1043580 |
| Plasma | Tissue and matrix | logFu | — no normalized value | — value does not convert to pX | Rattus norvegicus | CHEMBL1100461 |
| Plasma | Tissue and matrix | PPB | — no normalized value | — value does not convert to pX | Homo sapiens | CHEMBL4052363 |
| Plasma | Tissue and matrix | t1/2 | — no normalized value | — value does not convert to pX | Rattus norvegicus | CHEMBL3106283 |
| Plasma | Tissue and matrix | t1/2 | — no normalized value | — value does not convert to pX | Mus musculus | CHEMBL3106282 |
| Plasma | Tissue and matrix | Cp | — no normalized value | — value does not convert to pX | Rattus norvegicus | CHEMBL901030 |
| Plasma | Tissue and matrix | Drug uptake | — no normalized value | — value does not convert to pX | Rattus norvegicus | CHEMBL954089 |
| Plasma | Tissue and matrix | Stability | — no normalized value | — value does not convert to pX | Homo sapiens | CHEMBL2033724 |
| Plasma | Tissue and matrix | Cp | — no normalized value | — value does not convert to pX | Mus musculus | CHEMBL2156604 |
| Plasma | Tissue and matrix | Cp(f)max | — no normalized value | — value does not convert to pX | Rattus norvegicus | CHEMBL3111747 |