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TargetTissue and matrix

Liver microsome

Preparations such as liver microsomes or whole blood. Values below are reported as measured; because this is not a molecular target, they are not treated as affinities anywhere on this site.

Measurements
37
Compounds
3
Binding constants
0
Median pX
—

I · Identity

What this target is

Its function as UniProt states it, where in a cell the protein is found, and which cell types and tissues transcribe its gene.

Liver microsome has no protein record here. A name resolves when ChEMBL’s own target record gives an accession, when the name appears verbatim in a gene’s synonym list, or when it matches a UniProt protein name exactly. Guessing from a name that merely looks like a receptor is how a histone gene ends up filed as an adrenoceptor.

IV · Evidence

Every measurement at this target

Each row links to the ChEMBL assay it came from.

Other measurements 37

Everything else ChEMBL recorded for this compound — percentage inhibition, efficacy, half-life, cytotoxicity. Reported in the assay's own units, which is why no value is converted here.

TargetClassTypeValue (nM)pXOrganismAssay
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3540995
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3540994
Liver microsomeTissue and matrixKm— no normalized value— value does not convert to pXHomo sapiensCHEMBL3540992
Liver microsomeTissue and matrixVmax— no normalized value— value does not convert to pXHomo sapiensCHEMBL3540991
Liver microsomeTissue and matrixVmax— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538794
Liver microsomeTissue and matrixVmax— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538793
Liver microsomeTissue and matrixKm— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538786
Liver microsomeTissue and matrixKm— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538785
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538783
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538782
Liver microsomeTissue and matrixT1/2— no normalized value— value does not convert to pXHomo sapiensCHEMBL3637651
Liver microsomeTissue and matrixT1/2— no normalized value— value does not convert to pXHomo sapiensCHEMBL3637657
Liver microsomeTissue and matrixCLH— no normalized value— value does not convert to pXHomo sapiensCHEMBL3829956
Liver microsomeTissue and matrixT1/2— no normalized value— value does not convert to pXHomo sapiensCHEMBL3829950
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3540996
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3540993
Liver microsomeTissue and matrixDrug metabolism— no normalized value— value does not convert to pXHomo sapiensCHEMBL3537279
Liver microsomeTissue and matrixDrug metabolism— no normalized value— value does not convert to pXHomo sapiensCHEMBL3537278
Liver microsomeTissue and matrixDrug metabolism— no normalized value— value does not convert to pXHomo sapiensCHEMBL3537277
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538220
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538219
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538218
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538217
Liver microsomeTissue and matrixKm— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538216
Liver microsomeTissue and matrixVmax— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538215
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538214
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538213
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538212
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538211
Liver microsomeTissue and matrixKm— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538210
Liver microsomeTissue and matrixVmax— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538209
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538208
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538207
Liver microsomeTissue and matrixCL— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538206
Liver microsomeTissue and matrixFu— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538205
Liver microsomeTissue and matrixKm— no normalized value— value does not convert to pXHomo sapiensCHEMBL3538204
Liver microsomeTissue and matrixVmax— no normalized value— value does not convert to pXHomo sapiensCHEMBL3540997