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TargetUnclassified

HaCaT

Matched no rule. Shown as-is rather than assigned a class by guesswork. Values below are reported as measured; because this is not a molecular target, they are not treated as affinities anywhere on this site.

Measurements
41
Compounds
2
Binding constants
0
Median pX
—

I · Identity

What this target is

Its function as UniProt states it, where in a cell the protein is found, and which cell types and tissues transcribe its gene.

HaCaT has no protein record here. A name resolves when ChEMBL’s own target record gives an accession, when the name appears verbatim in a gene’s synonym list, or when it matches a UniProt protein name exactly. Guessing from a name that merely looks like a receptor is how a histone gene ends up filed as an adrenoceptor.

IV · Evidence

Every measurement at this target

Each row links to the ChEMBL assay it came from.

Functional readouts 1

IC₅₀, EC₅₀, AC₅₀ and potency. Assay-dependent, and not interchangeable with a binding constant.

TargetClassTypeValue (nM)pXOrganismAssay
HaCaTUnclassifiedIC50— no normalized value— value does not convert to pXHomo sapiensCHEMBL5577217

Other measurements 40

Everything else ChEMBL recorded for this compound — percentage inhibition, efficacy, half-life, cytotoxicity. Reported in the assay's own units, which is why no value is converted here.

TargetClassTypeValue (nM)pXOrganismAssay
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840386
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840387
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840388
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840389
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840390
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840391
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840392
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840393
HaCaTUnclassifiedFC— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840394
HaCaTUnclassifiedFC— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840395
HaCaTUnclassifiedFlu intensity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840396
HaCaTUnclassifiedFlu intensity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840397
HaCaTUnclassifiedFlu intensity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840398
HaCaTUnclassifiedFlu intensity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840399
HaCaTUnclassifiedFlu intensity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840400
HaCaTUnclassifiedFlu intensity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840401
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840406
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840407
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL4840408
HaCaTUnclassifiedInhibition— no normalized value— value does not convert to pXHomo sapiensCHEMBL5577216
HaCaTUnclassifiedInhibition— no normalized value— value does not convert to pXHomo sapiensCHEMBL5577216
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638409
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638410
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638411
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638412
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638413
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638414
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638415
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638416
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638417
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638421
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638422
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638423
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638424
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638425
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638426
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638427
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638428
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638430
HaCaTUnclassifiedActivity— no normalized value— value does not convert to pXHomo sapiensCHEMBL5638431