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TargetOrganisms

Cavia porcellus

Whole-organism screens (antiparasitic, antibacterial, antiviral). Values below are reported as measured; because this is not a molecular target, they are not treated as affinities anywhere on this site.

Measurements
59
Compounds
13
Binding constants
13
Median pX
—

I · Identity

What this target is

Its function as UniProt states it, where in a cell the protein is found, and which cell types and tissues transcribe its gene.

No single gene answers to Cavia porcellus. Names like this one are families or unsubtyped preparations — a measurement made against whatever receptors a tissue carried, before or without resolving which subtype bound the compound. A family has no one accession, and picking a member to stand for it would invent a precision the assay never had: asked for “Muscarinic acetylcholine receptor” UniProt returns CHRM1, and that answer is wrong.

Resolver said no gene lists this target name as a synonym — recorded by tools/fetch_expression.py, not written here.

IV · Evidence

Every measurement at this target

Each row links to the ChEMBL assay it came from.

Equilibrium binding constants 13

Ki and Kd — a concentration at equilibrium. Directly comparable across rows at the same target.

TargetClassTypeValue (nM)pXOrganismAssay
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL686245
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL686245
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL633438
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL633439
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL633440
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL683404
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL627982
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL627983
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL627984
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL627981
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL686245
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL693096
Cavia porcellusOrganismsKd— no normalized value— value does not convert to pXCavia porcellusCHEMBL693096

Functional readouts 6

IC₅₀, EC₅₀, AC₅₀ and potency. Assay-dependent, and not interchangeable with a binding constant.

TargetClassTypeValue (nM)pXOrganismAssay
Cavia porcellusOrganismsEC50— no normalized value— value does not convert to pXCavia porcellusCHEMBL858285
Cavia porcellusOrganismsEC50— no normalized value— value does not convert to pXCavia porcellusCHEMBL680361
Cavia porcellusOrganismsIC50— no normalized value— value does not convert to pXCavia porcellusCHEMBL692807
Cavia porcellusOrganismsEC50— no normalized value— value does not convert to pXCavia porcellusCHEMBL883445
Cavia porcellusOrganismsIC50— no normalized value— value does not convert to pXCavia porcellusCHEMBL686659
Cavia porcellusOrganismsIC50— no normalized value— value does not convert to pXCavia porcellusCHEMBL688857

Other measurements 40

Everything else ChEMBL recorded for this compound — percentage inhibition, efficacy, half-life, cytotoxicity. Reported in the assay's own units, which is why no value is converted here.

TargetClassTypeValue (nM)pXOrganismAssay
Cavia porcellusOrganismsContraction— no normalized value— value does not convert to pXCavia porcellusCHEMBL841378
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL687299
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL687299
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL687299
Cavia porcellusOrganismspKB— no normalized value— value does not convert to pXCavia porcellusCHEMBL696089
Cavia porcellusOrganismspKB— no normalized value— value does not convert to pXCavia porcellusCHEMBL696088
Cavia porcellusOrganismspKB— no normalized value— value does not convert to pXCavia porcellusCHEMBL880163
Cavia porcellusOrganismsED50— no normalized value— value does not convert to pXCavia porcellusCHEMBL681117
Cavia porcellusOrganismsED50— no normalized value— value does not convert to pXCavia porcellusCHEMBL681119
Cavia porcellusOrganismspD2— no normalized value— value does not convert to pXCavia porcellusCHEMBL841900
Cavia porcellusOrganismspD2— no normalized value— value does not convert to pXCavia porcellusCHEMBL841900
Cavia porcellusOrganismsRelative potency— no normalized value— value does not convert to pXCavia porcellusCHEMBL841375
Cavia porcellusOrganismsRelative potency— no normalized value— value does not convert to pXCavia porcellusCHEMBL841375
Cavia porcellusOrganismsRelative potency— no normalized value— value does not convert to pXCavia porcellusCHEMBL841375
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL818455
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL818455
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL818455
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL843391
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL843391
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL843391
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL843391
Cavia porcellusOrganismspD2— no normalized value— value does not convert to pXCavia porcellusCHEMBL842866
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL843381
Cavia porcellusOrganismsContraction— no normalized value— value does not convert to pXCavia porcellusCHEMBL841860
Cavia porcellusOrganismsContraction— no normalized value— value does not convert to pXCavia porcellusCHEMBL841863
Cavia porcellusOrganismsContraction— no normalized value— value does not convert to pXCavia porcellusCHEMBL842626
Cavia porcellusOrganismsContraction— no normalized value— value does not convert to pXCavia porcellusCHEMBL841861
Cavia porcellusOrganismsContraction— no normalized value— value does not convert to pXCavia porcellusCHEMBL842627
Cavia porcellusOrganismsContraction— no normalized value— value does not convert to pXCavia porcellusCHEMBL841862
Cavia porcellusOrganismsED50— no normalized value— value does not convert to pXCavia porcellusCHEMBL685644
Cavia porcellusOrganismsED50— no normalized value— value does not convert to pXCavia porcellusCHEMBL684863
Cavia porcellusOrganismsInhibition— no normalized value— value does not convert to pXCavia porcellusCHEMBL688147
Cavia porcellusOrganismspD2— no normalized value— value does not convert to pXCavia porcellusCHEMBL688171
Cavia porcellusOrganismsEfficacy— no normalized value— value does not convert to pXCavia porcellusCHEMBL686257
Cavia porcellusOrganismsLog B/F— no normalized value— value does not convert to pXCavia porcellusCHEMBL683300
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL687000
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL686990
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL686990
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL686991
Cavia porcellusOrganismsKb— no normalized value— value does not convert to pXCavia porcellusCHEMBL686991
Cavia porcellus · Psychedelia